16,040
回編集
「P2Y受容体」の版間の差分
細
→P2Y14受容体
細 (→P2Y14受容体) |
細 (→P2Y14受容体) |
||
| 66行目: | 66行目: | ||
|- | |- | ||
| [[P2RY1|P2RY<sub>1</sub>]] || {{Gene|P2RY1}} || G<sub>q/11</sub> ||2MeSADP <br>MRS2365 <br>compound 3a <br>ADPβS <br>2',3'-ddATP <br>dATPαS <br>ATPγS <br>2MeSATP <br>ATP <br>ADP ||MRS2500<br>MRS2279 <br>MRS2298 <br>MRS2496<br> | | [[P2RY1|P2RY<sub>1</sub>]] || {{Gene|P2RY1}} || G<sub>q/11</sub> ||2MeSADP <br>MRS2365 <br>compound 3a <br>ADPβS <br>2',3'-ddATP <br>dATPαS <br>ATPγS <br>2MeSATP <br>ATP <br>ADP ||MRS2500<br>MRS2279 <br>MRS2298 <br>MRS2496<br> | ||
MRS2179 <br>MRS2950 <br>2,2'-pyridylisatogen tosylate <br>2-ClATP <br>suramin <br>2MeSATP <br>PPADS <br>ATP <br>A2P5P <br>adenosine-3'-5'-bisphosphate | MRS2179 <br>MRS2950 <br>2,2'-pyridylisatogen tosylate <br>2-ClATP <br>suramin <br>2MeSATP <br>PPADS <br>ATP <br>A2P5P <br>adenosine-3'-5'-bisphosphate | ||
|- | |- | ||
| [[P2RY2|P2RY<sub>2</sub>]] || {{Gene|P2RY2}} || G<sub>q/11</sub> ||MRS2698 <br>UTP <br>4-thio-UTP <br>2-thioUTP <br>ATP <br>diquafosol <br>PSB1114 <br>denufosol <br>Ap4A <br>UTPγS <br>5BrUTP <br>MRS2768||AR-C126313 <br>AR-C118925XX <br>reactive blue-2 <br>suramin | | [[P2RY2|P2RY<sub>2</sub>]] || {{Gene|P2RY2}} || G<sub>q/11</sub> ||MRS2698 <br>UTP <br>4-thio-UTP <br>2-thioUTP <br>ATP <br>diquafosol <br>PSB1114 <br>denufosol <br>Ap4A <br>UTPγS <br>5BrUTP <br>MRS2768||AR-C126313 <br>AR-C118925XX <br>reactive blue-2 <br>suramin | ||
| 84行目: | 83行目: | ||
|} | |} | ||
編集部にて[[w:P2Y purinergic receptor|Wikipedia]]より翻訳、改変。 | 編集部にて[[w:P2Y purinergic receptor|Wikipedia]]より翻訳、改変。 | ||
{| class="wikitable" | |||
|+表2. P2Y受容体 | |||
|- | |||
!受容体!!内在性アゴニスト!!アゴニスト!!選択的アゴニスト!!アンタゴニスト | |||
|- | |||
| P2Y1||ADP>ATP||ADPβS<br>2MeSADP||MRS2365<br>2-Cl-ADP (α-BH3)||MRS2500<br>BMS compound 16<br>MRS2279<br>MRS2179<br>2‐2'‐ピリジルイサトゲントシラート | |||
|- | |||
| P2Y2||UTP=ATP||||2-thioUTP<br>PSB1114<br>Ap4A<br>UTPγS<br>MRS2768||AR-C118925XX | |||
|- | |||
| P2Y4||UTPe>ATP||||MRS4062<br>UTPγS||ATP (ヒト受容体） | |||
|- | |||
| P2Y6||UDP>>UTP>ATP||Rp-5-OMe-UDPαB||MRS295MRS2693<br>3-phenacyl-UDP7||MRS2578 | |||
|- | |||
| P2Y11||ATP>UTP||AR-C67085<br>NF546<br>NAADP<br>NAD||NF340||NF157 | |||
|- | |||
| P2Y12||ADP||2MeSADP||||PSB-0739<br>AZD1283<br>チカグレロル<br>ARL66096 | |||
|- | |||
| P2Y13||ADP>>ATP||||||MRS2211 | |||
|- | |||
| P2Y14||UDP ≥ UDP-glucose||MRS2690||||PPTN | |||
|} | |||
== 参考文献 == | == 参考文献 == | ||
<references /> | <references /> | ||